0
Correspondence |

Evaluation of the Penetration of Fluoroquinolones in Human Conjunctival Tissue—Reply

Rudolph S. Wagner, MD
[+] Author Affiliations

Copyright 2006 American Medical Association. All Rights Reserved. Applicable FARS/DFARS Restrictions Apply to Government Use.

More Author Information
Arch Ophthalmol. 2006;124(12):1797-1797. doi:10.1001/archopht.124.12.1797-a
Text Size: A A A
Published online

In reply

We appreciate the comments from Drs Fiscella and Jensen. The dual-biopsy technique is an optimal method for assessing conjunctival anti-infective concentrations. And, we strongly agree that additional factors should also be considered when evaluating drug efficacy.

Conjunctival drug levels are of particular importance in bacterial conjunctivitis because the conjunctiva is the tissue to which the bacteria adhere—the site of infection. This, of course, is not a difficult concept. We disagree that the formulation concentration differences between 0.5% moxifloxacin and 0.3% gatifloxacin resulted in the difference in conjunctival concentration. In fact, 0.5% levofloxacin had a lower mean conjunctival concentration (2.34 μg/g) than 0.3% gatifloxacin (2.54 μg/g).

The dual-biopsy technique is an excellent method for measuring anti-infective drug concentrations and could also be adapted for any other ophthalmic medication. To obtain an adequate quantity of tissue for analysis, previous methods for assessing conjunctival antibiotic concentrations described 1 large biopsy specimen taken during cataract surgery.1 Our method uses 2 smaller tissue samples that can be taken in the office in a normal patient population. This allows for rapid healing and less chance of infection.

We agree that gatifloxacin may be a choice superior to ciprofloxacin in treating ocular infection. The same can be said of moxifloxacin, a fourth-generation fluoroquinolone like gatifloxacin that also offers lower minimum inhibitory concentrations and may be less susceptible to resistance compared with previous fluoroquinolone generations.2

There is no clinical evidence of any safety issues with any of the fluoroquinolones studied. The moxifloxacin Food and Drug Administration labeling states that ocular adverse events were reported in approximately 1% to 6% of subjects while the gatifloxacin Food and Drug Administration labeling states that some ocular adverse events were seen at a rate of 5% to 10%. We are very fortunate to have exceptional safety profiles for all of the leading ophthalmic antibiotics. We agree that gatifloxacin, which is indicated to be dosed at a higher frequency than moxifloxacin (every 2 hours for up to 8 times daily on days 1 and 2), is an entirely safe and effective medication.

The referenced studies do not meet the standards of well-controlled clinical trials. Certainly, the “open-label, partially randomized” study performed by Moshirfar et al3 requires no further comment. It is also important to note that 2 separate groups4 5 were unable to reproduce the results found by Solomon et al.6 In addition, Donnenfeld et al7 reported major end points graded using scales that were “not validated or standardized.” In any case, this is not the forum for discussing corneal wound healing studies when the subject at hand is bacterial conjunctivitis.

Last, it should be noted that following the biopsy procedure, all of the subjects were provided with moxifloxacin to be used prophylactically for 1 week. Subjects were seen at 1 day and 1 week after the biopsy to monitor healing, and no subjects in our study evidenced a delay in wound healing.

AUTHOR INFORMATION

Correspondence: Dr Wagner, Doctors Office Center, Suite 6100, PO Box 1709, Newark, NJ 07101-1709 (wagdoc@comcast.net).

Financial Disclosure: None reported.

REFERENCES

Tabbara  KF, al-Kharashi  SA, al-Mansouri  SM.  et al.  Ocular levels of azithromycin. Arch Ophthalmol 1998;1161625- 1628
PubMed
Mah  FS. Fourth-generation fluoroquinolones: new topical agents in the war on ocular bacterial infections. Curr Opin Ophthalmol 2004;15316- 320
PubMed
Moshirfar  M, Marx  DP, Kumar  R. The effect of the fourth-generation fluoroquinolones on corneal reepithelialization after penetrating keratoplasty. Cornea 2005;24833- 836
PubMed
Setabutr  P, Sami  MS, Folterman  MO, Chuang  AZ, Yee  RW. A comparison of epithelial healing rates with topical moxifloxacin and gatifloxacin after bilateral photorefractive keratectomy (PRK) [ARVO abstract]. Invest Ophthalmol Vis Sci 2005;46E-abstract 4878See abstracthereAccessed June 6, 2006
Burka  JM, Bower  KS, VanRoekel  RC, Stutzman  RD, Kuzmowych  CP, Howard  RH. The effect of fourth-generation fluoroquinolones gatifloxacin and moxifloxacin on epithelial healing following photorefractive keratectomy. Am J Ophthalmol 2005;14083- 87
PubMed
Solomon  R, Donnenfeld  ED, Wittpenn  JR.  et al.  Effect of gatifloxacin 0.3% and moxifloxacin 0.5% on corneal epithelial wound healing after photorefractive keratectomy.  Presented at: 2005 Association for Research in Vision and Ophthalmology Annual Meeting May 5, 2005 Fort Lauderdale, Fla
Donnenfeld  E, Perry  HD, Chruscicki  DA, Bitterman  A, Cohn  S, Solomon  R. A comparison of the fourth-generation fluoroquinolones gatifloxacin 0.3% and moxifloxacin 0.5% in terms of ocular tolerability. Curr Med Res Opin 2004;201753- 1758
PubMed

First Page Preview

First page PDF preview

Figures

Tables

Interactive Graphics

Video

Country-Specific Mortality and Growth Failure in Infancy and Yound Children and Association With Material Stature

Use interactive graphics and maps to view and sort country-specific infant and early dhildhood mortality and growth failure data and their association with maternal

Tabbara  KF, al-Kharashi  SA, al-Mansouri  SM.  et al.  Ocular levels of azithromycin. Arch Ophthalmol 1998;1161625- 1628
PubMed
Mah  FS. Fourth-generation fluoroquinolones: new topical agents in the war on ocular bacterial infections. Curr Opin Ophthalmol 2004;15316- 320
PubMed
Moshirfar  M, Marx  DP, Kumar  R. The effect of the fourth-generation fluoroquinolones on corneal reepithelialization after penetrating keratoplasty. Cornea 2005;24833- 836
PubMed
Setabutr  P, Sami  MS, Folterman  MO, Chuang  AZ, Yee  RW. A comparison of epithelial healing rates with topical moxifloxacin and gatifloxacin after bilateral photorefractive keratectomy (PRK) [ARVO abstract]. Invest Ophthalmol Vis Sci 2005;46E-abstract 4878See abstracthereAccessed June 6, 2006
Burka  JM, Bower  KS, VanRoekel  RC, Stutzman  RD, Kuzmowych  CP, Howard  RH. The effect of fourth-generation fluoroquinolones gatifloxacin and moxifloxacin on epithelial healing following photorefractive keratectomy. Am J Ophthalmol 2005;14083- 87
PubMed
Solomon  R, Donnenfeld  ED, Wittpenn  JR.  et al.  Effect of gatifloxacin 0.3% and moxifloxacin 0.5% on corneal epithelial wound healing after photorefractive keratectomy.  Presented at: 2005 Association for Research in Vision and Ophthalmology Annual Meeting May 5, 2005 Fort Lauderdale, Fla
Donnenfeld  E, Perry  HD, Chruscicki  DA, Bitterman  A, Cohn  S, Solomon  R. A comparison of the fourth-generation fluoroquinolones gatifloxacin 0.3% and moxifloxacin 0.5% in terms of ocular tolerability. Curr Med Res Opin 2004;201753- 1758
PubMed

Correspondence

CME Course for:


You need to register in order to view this quiz.


To understand the clinical management of acute heart failure syndromes.
Accreditation Information The American Medical Association is accredited by the Accreditation Council for Continuing Medical Education to provide continuing medical education for physicians.
The AMA designates this journal-based CME activity for a maximum of 1 AMA PRA Category 1 CreditTM per course. Physicians should claim only the credit commensurate with the extent of their participation in the activity.
Physicians who complete the CME course and score at least 80% correct on the quiz are eligible for AMA PRA Category 1 CreditTM.
Note: You must get at least of the answers correct to pass this quiz.
Note: You must get at least of the answers correct to pass this quiz.
You have not filled in all the answers to complete this quiz
The following questions were not answered:
Sorry, you have unsuccessfully completed this CME quiz with a score of
The following questions were not answered correctly:
For CME Course: A Proposed Model for Initial Assessment and Management of Acute Heart Failure Syndromes
Indicate what changes(s) you will implement in your practice, if any, based on this CME course.
To view and print your certificate and access a summary of your CME courses go to My CME.
NOTE:
Citing articles are presented as examples only. In non-demo SCM6 implementation, integration with CrossRef’s “Cited By” API will populate this tab (http://www.crossref.org/citedby.html).
Submit a Comment

Some tools below are only available to our subscribers or users with an online account.

Related Content

Customize your page view by dragging & repositioning the boxes below.

See Also...
Articles Related By Topic
Related Topics
PubMed Articles